SCHEMBL4693261

SCHEMBL4693261

COc1ccccc1C(=O)N1CC2CN(CC[C@H](N)c3ccccc3)CC2C1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 6/20 0.51
HCRTR2 O43614 6/20 0.51
POLB P06746 1/20 0.49
GAA P10253 1/20 0.49
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPK14 Q16539 1/20 0.47
CCR5 P51681 3/20 0.46
HTT P42858 1/20 0.46
KCNK3 O14649 2/20 0.46
KCNK9 Q9NPC2 2/20 0.46
DRD3 P35462 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695959 0.88 HCRTR2 (0.53) HCRTR1HCRTR2GAACCR5KCNK3
SCHEMBL4691899 0.88 CCR5 (0.43) HCRTR1HCRTR2CCR5
SCHEMBL4694065 0.86 CCR5 (0.52) HCRTR1HCRTR2CCR5
SCHEMBL4690615 0.86 HCRTR1 (0.52) HCRTR1HCRTR2CCR5
SCHEMBL4695358 0.86 GAA (0.57) HCRTR1HCRTR2GAAALDH1A1KDM4E
SCHEMBL4695158 0.85 CCR5 (0.55) HCRTR1HCRTR2CCR5
SCHEMBL4695827 0.85 HCRTR1 (0.46) HCRTR1HCRTR2GAAALDH1A1CCR5
SCHEMBL4690598 0.84 CCR5 (0.55) HCRTR1HCRTR2CCR5
SCHEMBL4690143 0.83 MAPK14 (0.52) HCRTR1HCRTR2ALDH1A1MAPK14CCR5
SCHEMBL4689905 0.83 CCR5 (0.52) POLBCYP2C9CYP2C19MAPK14CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed