SCHEMBL4693306

SCHEMBL4693306

O=C1CCc2cccc(Cl)c2N1Cc1cc(Cl)cc(N2CCNCC2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 2/20 0.44
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
HTR6 P50406 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
HTR2C P28335 2/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
TP53 P04637 1/20 0.43
CYP3A4 P08684 1/20 0.43
HTR1A P08908 1/20 0.43
CYP2D6 P10635 1/20 0.43
THRB P10828 1/20 0.43
HTR2A P28223 1/20 0.43
SLC6A4 P31645 1/20 0.43
HTR7 P34969 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4486014 0.85 POLB (0.57) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL4493695 0.81 HDAC1 (0.54) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL3324240 0.78 HTR6 (0.60) ADRB1HTR6HTR3EHTR3BHTR1A
SCHEMBL4468502 0.73 POLB (0.60) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL4492877 0.73 POLB (0.53) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL4483596 0.73 POLB (0.53) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL4558610 0.73 POLB (0.50) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL4464670 0.72 POLB (0.51) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL4480619 0.70 POLB (0.49) ADRB1CHRM2CHRM4CHRM1CHRM3
SCHEMBL31430299 0.70 CHRM5 (0.58) GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603880-B1 QUINOLINONE/BENZOXAZINONE DERIVATIVES AND USES THEREOF HOFFMANN LA ROCHE (CH) 2008-05-07 EP claimed