SCHEMBL4693979

SCHEMBL4693979

Nc1nc(N)c2c(cc(-c3ccccc3C(F)(F)F)c3c2ccn3CC(O)C(F)(F)C(=O)OF)n1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 9/20 0.35
PAX8 Q06710 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
PTPN1 P18031 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691391 0.83 SLC2A1 (0.36) SLC2A1PAX8GRIN1GRIN2BPTPN1
SCHEMBL4689868 0.82 SLC2A1 (0.41) SLC2A1PAX8GRIN1GRIN2BPTPN1
SCHEMBL4691192 0.82 GRIN1 (0.36) SLC2A1PAX8GRIN1GRIN2BPTPN1
SCHEMBL4688933 0.80 SLC2A1 (0.40) SLC2A1PTPN1
Trifluoroacetic Acid SCHEMBL4691189 0.80 SLC2A1 (0.39) SLC2A1PAX8GRIN1GRIN2BPTPN1
Trifluoroacetic Acid SCHEMBL4691388 0.79 SCN5A (0.38) SLC2A1PAX8GRIN1GRIN2BPTPN1
Trifluoroacetic Acid SCHEMBL4690935 0.77 SLC2A1 (0.39) SLC2A1PAX8GRIN1GRIN2BPTPN1
SCHEMBL4688280 0.76 SLC2A1 (0.42) SLC2A1PAX8
SCHEMBL4687979 0.75 DHFR (0.46) SLC2A1PTPN1
SCHEMBL4710085 0.73 GRIN2B (0.38) GRIN1GRIN2BPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1628979-B1 DIAMINOPYRROLOQUINAZOLINES COMPOUNDS AS PROTEIN TYROSINE PHOSPHATASE INHIBITORS HOFFMANN LA ROCHE (CH) 2008-03-19 EP disclosed