SCHEMBL4694069

SCHEMBL4694069

Cc1ccc(N(CCCN2CC3CN(C(=O)c4c(C)ccnc4C)CC3C2)C(=O)Nc2ccc(OC(F)(F)F)cc2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 12/20 0.40
MCHR1 Q99705 1/20 0.38
EPHX2 P34913 1/20 0.37
MAPT P10636 1/20 0.37
MEN1 O00255 1/20 0.36
TP53 P04637 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
KCNH2 Q12809 1/20 0.36
ABL1 P00519 1/20 0.36
TRPV1 Q8NER1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695550 0.92 CCR5 (0.41) CCR5MCHR1KCNH2
SCHEMBL4690299 0.91 CCR5 (0.41) CCR5EPHX2KCNH2
SCHEMBL4690734 0.90 KCNH2 (0.45) CCR5KCNH2
SCHEMBL4690606 0.90 CCR5 (0.42) CCR5EPHX2MAPTMEN1KMT2A
SCHEMBL4690440 0.90 CCR5 (0.42) CCR5EPHX2KCNH2
SCHEMBL4694144 0.90 CCR5 (0.42) CCR5EPHX2MAPTKCNH2
SCHEMBL4694951 0.89 CCR5 (0.48) CCR5
SCHEMBL4691634 0.88 CCR5 (0.42) CCR5MCHR1KCNH2
SCHEMBL4695270 0.88 CCR5 (0.41) CCR5EPHX2KCNH2
SCHEMBL4690519 0.88 CCR5 (0.41) CCR5EPHX2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed