SCHEMBL4694199

SCHEMBL4694199

Nc1cnc(Br)c(-c2ccncc2Cl)n1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
LIMK1 P53667 1/20 0.40
IDO1 P14902 1/20 0.38
ADORA2B P29275 5/20 0.37
ADORA2A P29274 5/20 0.37
NQO2 P16083 3/20 0.37
NFATC1 O95644 1/20 0.36
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
CDC25B P30305 1/20 0.35
SCN2A Q99250 1/20 0.35
CCNC P24863 1/20 0.34
CDK8 P49336 1/20 0.34
LATS1 O95835 3/20 0.33
KCNH2 Q12809 1/20 0.33
AOC3 Q16853 1/20 0.33
IMPDH2 P12268 2/20 0.33
LATS2 Q9NRM7 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3063403 0.81 GAA (0.44) GAALIMK1IDO1ADORA2BADORA2A
SCHEMBL14545378 0.78 ADORA2A (0.45) GAALIMK1ADORA2BADORA2ANQO2
SCHEMBL3063962 0.77 ADORA2B (0.57) LIMK1ADORA2BADORA2ANQO2
SCHEMBL4690211 0.73 CNR1 (0.60) ADORA2BADORA2ANQO2
SCHEMBL3077195 0.72 ADORA2A (0.45) ADORA2BADORA2ANQO2
SCHEMBL3066532 0.71 ADORA2B (0.55) ADORA2BADORA2ANQO2
SCHEMBL4693972 0.70 GAA (0.47) GAALIMK1IDO1ADORA2BADORA2A
SCHEMBL18039071 0.69 ADORA2B (0.51) GAALIMK1IDO1ADORA2BADORA2A
SCHEMBL31301252 0.69 GSK3B (0.59) GAALIMK1IDO1NFATC1GSK3B
SCHEMBL1975440 0.67 GAA (0.47) GAALIMK1ADORA2BADORA2ANQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871762-A2 SUBTITUTED HETEROARYL CB1 ANTAGONISTS NEUROGEN CORPORATION (US) 2008-01-02 EP disclosed
US-20070078135-A1 Substituted heteroaryl CB1 antagonists NEUROGEN CORPORATION (US) 2007-04-05 US disclosed
US-20070078135-A1 Substituted heteroaryl CB1 antagonists NEUROGEN CORPORATION (US) 2007-04-05 US disclosed
US-20070078135-A1 Substituted heteroaryl CB1 antagonists NEUROGEN CORPORATION (US) 2007-04-05 US disclosed
WO-2006113704-A2 SUBTITUTED HETEROARYL CB1 ANTAGONISTS NEUROGEN CORPORATION (US) 2006-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070078135-A1 Substituted heteroaryl CB1 antagonists CNR1, CNR2, OPRL1 GAA 1332/4885LIMK1 4710/4885IDO1 764/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.