SCHEMBL4694346

SCHEMBL4694346

COc1ccc(F)cc1C(=O)N1CC2CN(CCC(=O)Nc3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
MAPT P10636 4/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
TSHR P16473 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
KCNK3 O14649 2/20 0.46
KCNK9 Q9NPC2 2/20 0.46
LMNA P02545 2/20 0.45
GAA P10253 2/20 0.45
ALDH1A1 P00352 1/20 0.45
MEN1 O00255 1/20 0.43
PKM P14618 1/20 0.43
BLM P54132 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692701 0.91 CYP2C9 (0.51) KMT2ASMN1; SMN2MAPTCYP1A2CYP3A4
SCHEMBL4691831 0.91 MAPT (0.51) KMT2ASMN1; SMN2MAPTTSHRCYP1A2
SCHEMBL4691400 0.91 KMT2A (0.50) KMT2AMAPTTSHRKCNK3KCNK9
SCHEMBL4692708 0.90 CYP1A2 (0.49) KMT2ASMN1; SMN2MAPTCYP1A2CYP3A4
SCHEMBL4692942 0.88 CYP2C9 (0.49) KMT2ASMN1; SMN2MAPTCYP1A2CYP3A4
SCHEMBL4694353 0.87 KCNK3 (0.46) KMT2ASMN1; SMN2MAPTL3MBTL1TSHR
SCHEMBL4693950 0.87 HCRTR1 (0.49) KMT2ASMN1; SMN2MAPTCYP1A2CYP3A4
SCHEMBL4692624 0.86 HCRTR1 (0.50) KMT2ASMN1; SMN2MAPTLMNAALDH1A1
SCHEMBL4693167 0.86 HCRTR1 (0.50) KMT2ASMN1; SMN2MAPTCYP1A2CYP3A4
SCHEMBL4693892 0.86 HCRTR1 (0.47) KMT2ASMN1; SMN2MAPTTSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed