SCHEMBL4694353

SCHEMBL4694353

COc1ccc(F)cc1C(=O)N1CC2CN(CCCNc3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 3/20 0.46
KCNK9 Q9NPC2 3/20 0.46
GFER P55789 1/20 0.44
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HCRTR1 O43613 3/20 0.41
HCRTR2 O43614 3/20 0.41
GAA P10253 2/20 0.41
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
DUSP3 P51452 1/20 0.39
PTPN5 P54829 1/20 0.39
PTPN11 Q06124 1/20 0.39
EPHA2 P29317 1/20 0.39
KDR P35968 1/20 0.39
EPHB4 P54760 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691874 0.92 ALDH1A1 (0.43) KCNK3KCNK9HCRTR1HCRTR2GAA
SCHEMBL4691840 0.92 MAPT (0.47) GFERSMN1; SMN2HCRTR1HCRTR2GAA
SCHEMBL4691406 0.91 HCRTR1 (0.48) KCNK3KCNK9KMT2AHCRTR1HCRTR2
SCHEMBL4692704 0.91 HCRTR1 (0.49) KCNK3KCNK9SMN1; SMN2HCRTR1HCRTR2
SCHEMBL4692715 0.89 HCRTR1 (0.43) KCNK3KCNK9KMT2ASMN1; SMN2HCRTR1
SCHEMBL4694435 0.88 P2RX7 (0.47) KCNK3KCNK9KMT2ASMN1; SMN2HCRTR1
SCHEMBL4693956 0.88 HCRTR1 (0.49) KCNK3KCNK9KMT2ASMN1; SMN2HCRTR1
SCHEMBL4692947 0.88 CPS1 (0.41) KCNK3KCNK9SMN1; SMN2HCRTR1HCRTR2
SCHEMBL4692628 0.87 HCRTR1 (0.50) SMN1; SMN2HCRTR1HCRTR2GAAALDH1A1
SCHEMBL4694346 0.87 KMT2A (0.50) KCNK3KCNK9KMT2ASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed