SCHEMBL4694577

SCHEMBL4694577

CCCc1cc(CC(C)(CC(=O)N2CCC(C(=O)O)CC2)SN=O)c(C)cc1OCCN(C)C

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
ITGB3 P05106 1/20 0.31
ITGA2B P08514 1/20 0.31
RCE1 Q9Y256 2/20 0.31
ERBB2 P04626 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696863 0.86 MEN1 (0.37) MEN1KMT2ATSHRSMN1; SMN2RXFP1
SCHEMBL4693660 0.86 BDKRB1 (0.34) MEN1KMT2ATSHRSMN1; SMN2RXFP1
SCHEMBL6416941 0.80 SMN1; SMN2 (0.37) MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL6413365 0.74 TSHR (0.40) MEN1KMT2ATSHRSMN1; SMN2RXFP1
Hydrochloric Acid SCHEMBL4697561 0.69 SMN1; SMN2 (0.44) SMN1; SMN2
SCHEMBL4694686 0.69 CYP1A2 (0.35) MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL4694575 0.68 CYP1A2 (0.52) MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL6420748 0.65 CYP1A2 (0.33) SMN1; SMN2
SCHEMBL4692851 0.64 CYP1A2 (0.38) SMN1; SMN2
SCHEMBL4694902 0.64 CYP1A2 (0.38) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109542-A4 NITROSATED AND NITROSYLATED ALPHA-ADRENERGIC RECEPTOR ANTAGONISTS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-03-26 EP disclosed
EP-1109542-A1 NITROSATED AND NITROSYLATED ALPHA-ADRENERGIC RECEPTOR ANTAGONISTS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2001-06-27 EP disclosed
WO-2000012075-A1 NITROSATED AND NITROSYLATED ALPHA-ADRENERGIC RECEPTOR ANTAGONISTS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2000-03-09 WO disclosed