SCHEMBL4693660

SCHEMBL4693660

CCCc1cc(CC(C)(CC(=O)N2CCC(C(=O)O)CC2)Sc2c(OC)cc(OC)cc2OC)c(C)cc1OCCN(C)C

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 4/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
POLB P06746 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34
ERBB2 P04626 2/20 0.32
ELANE P08246 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
EPHX2 P34913 1/20 0.32
GAA P10253 1/20 0.32
TSHR P16473 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694577 0.86 MEN1 (0.35) MEN1KMT2ARXFP1ERBB2SMN1; SMN2
SCHEMBL4696863 0.83 MEN1 (0.37) MEN1KMT2APOLBRXFP1ERBB2
SCHEMBL4697597 0.74 GAA (0.44) MEN1KMT2APOLBRXFP1EPHX2
SCHEMBL4693654 0.71 CYP1A2 (0.47) BDKRB1MEN1KMT2APOLBSMN1; SMN2
SCHEMBL6413365 0.71 TSHR (0.40) MEN1KMT2APOLBRXFP1SMN1; SMN2
SCHEMBL6416941 0.70 SMN1; SMN2 (0.37) MEN1KMT2APOLBSMN1; SMN2GAA
SCHEMBL4696776 0.67 ALDH1A1 (0.53) MEN1KMT2APOLBSMN1; SMN2GAA
SCHEMBL4696088 0.62 ADRA1D (0.58) SMN1; SMN2GAA
SCHEMBL4695768 0.60 CYP1A2 (0.47) SMN1; SMN2GAALMNA
SCHEMBL6417121 0.60 ESR1 (0.52) SMN1; SMN2GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109542-A4 NITROSATED AND NITROSYLATED ALPHA-ADRENERGIC RECEPTOR ANTAGONISTS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-03-26 EP disclosed
EP-1109542-A1 NITROSATED AND NITROSYLATED ALPHA-ADRENERGIC RECEPTOR ANTAGONISTS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2001-06-27 EP disclosed
WO-2000012075-A1 NITROSATED AND NITROSYLATED ALPHA-ADRENERGIC RECEPTOR ANTAGONISTS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2000-03-09 WO disclosed