SCHEMBL4695342

SCHEMBL4695342

CC(c1ccccc1)C(CN)c1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.72
SLC6A4 P31645 6/20 0.55
SLC6A3 Q01959 6/20 0.55
SLC6A2 P23975 5/20 0.55
HTR2A P28223 2/20 0.52
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
HRH1 P35367 1/20 0.43
AOC3 Q16853 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
KCNH2 Q12809 2/20 0.41
ADRA2A P08913 1/20 0.40
ADRA2C P18825 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4692562 0.89 TAAR1 (0.58) TAAR1SLC6A4SLC6A3SLC6A2HTR2A
Hydrochloric Acid SCHEMBL5200363 0.87 TAAR1 (0.56) TAAR1SLC6A4SLC6A3SLC6A2HTR2A
SCHEMBL247628 0.84 TAAR1 (1.00) TAAR1SLC6A4SLC6A3SLC6A2HTR2A
SCHEMBL5005843 0.84 TAAR1 (1.00) TAAR1SLC6A4SLC6A3SLC6A2HTR2A
SCHEMBL5351663 0.84 TAAR1 (1.00) TAAR1SLC6A4SLC6A3SLC6A2HTR2A
SCHEMBL8995001 0.83 TAAR1 (0.73) TAAR1SLC6A4SLC6A3SLC6A2HTR2A
Hydrochloric Acid SCHEMBL1669712 0.82 TAAR1 (0.95) TAAR1SLC6A4SLC6A3SLC6A2HTR2A
SCHEMBL3729576 0.82 SLC6A2 (0.67) TAAR1SLC6A4SLC6A3SLC6A2CYP3A4
SCHEMBL12122150 0.81 TAAR1 (0.64) TAAR1SLC6A4SLC6A3SLC6A2HTR2A
SCHEMBL8953218 0.80 TAAR1 (0.69) TAAR1SLC6A4SLC6A3SLC6A2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP disclosed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2004048317-A1 SUBSTITUTED AMIDES ACTIVE AT THE CANNABINOID-1 RECEPTOR MERCK & CO., INC. (US) 2004-06-10 WO disclosed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO disclosed