SCHEMBL4695564

SCHEMBL4695564

O=C(CCc1cnc[nH]1)N[C@@H](CCN1CC2=CN(C(=O)c3c(F)cccc3Cl)CC2C1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 2/20 0.42
ICAM1 P05362 2/20 0.42
ITGAL P20701 2/20 0.42
CCR5 P51681 5/20 0.38
CYP19A1 P11511 2/20 0.34
SIGMAR1 Q99720 1/20 0.33
HRH2 P25021 1/20 0.32
HRH4 Q9H3N8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692079 0.87 CCR5 (0.44) ITGB2ICAM1ITGALCCR5SIGMAR1
SCHEMBL4689803 0.87 CCR5 (0.39) CCR5
SCHEMBL4692081 0.87 CCR5 (0.39) CCR5SIGMAR1
SCHEMBL4690183 0.85 CCR5 (0.43) CCR5SIGMAR1
SCHEMBL4695466 0.85 CCR5 (0.55) ITGB2ICAM1ITGALCCR5
SCHEMBL4695562 0.85 CCR5 (0.55) ITGB2ICAM1ITGALCCR5
SCHEMBL4691520 0.85 CCR5 (0.42) ITGB2ICAM1ITGALCCR5SIGMAR1
SCHEMBL4696260 0.84 CCR5 (0.40) CCR5SIGMAR1
SCHEMBL4691817 0.84 CCR5 (0.40) CCR5SIGMAR1
SCHEMBL4695068 0.84 CCR5 (0.44) ITGB2ICAM1ITGALCCR5SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed