SCHEMBL4695591

SCHEMBL4695591

O=C(O)C1c2c(cnn2CCc2ccccc2)C2CN1C(=O)N2O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 1/20 0.33
S1PR1 P21453 1/20 0.33
S1PR5 Q9H228 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GAA P10253 2/20 0.33
HTT P42858 2/20 0.33
USP2 O75604 1/20 0.33
MAPT P10636 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
AADAT Q8N5Z0 1/20 0.32
GRN P28799 1/20 0.32
SORT1 Q99523 1/20 0.32
TP53 P04637 1/20 0.31
POLB P06746 1/20 0.31
MAPK1 P28482 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695590 1.00 PFKFB3 (0.33) PFKFB3S1PR1S1PR5MEN1KMT2A
SCHEMBL4142503 0.89 POLB (0.37) MAPTL3MBTL1NPC1RAB9ASMN1; SMN2
SCHEMBL4697841 0.85 KCNA5 (0.32) PFKFB3S1PR1S1PR5MEN1KMT2A
SCHEMBL4697845 0.85 KCNA5 (0.32) PFKFB3S1PR1S1PR5MEN1KMT2A
SCHEMBL4695501 0.83 MEN1 (0.31) PFKFB3MEN1KMT2ASMN1; SMN2
SCHEMBL4695499 0.83 MEN1 (0.31) PFKFB3MEN1KMT2ASMN1; SMN2
SCHEMBL4696935 0.83 MEN1 (0.31) PFKFB3MEN1KMT2ASMN1; SMN2
SCHEMBL5254763 0.82
SCHEMBL20557430 0.78 KDM4E (0.30) GAA
SCHEMBL20557547 0.78 KCNA5 (0.33) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed