SCHEMBL4696115

SCHEMBL4696115

COc1cccc(C(=O)N2CC3CN(CCCN(C(=O)OC4CCN(C(C)=O)CC4)c4ccc(C)c(Cl)c4)CC3C2)c1OC

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.47
CCR5 P51681 17/20 0.46
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693851 0.96 KCNH2 (0.48) KCNH2CCR5
SCHEMBL4691237 0.94 KCNH2 (0.47) KCNH2CCR5HCRTR1HCRTR2
SCHEMBL4695409 0.94 CCR5 (0.49) KCNH2CCR5
SCHEMBL4694016 0.93 KCNH2 (0.46) KCNH2CCR5
SCHEMBL4691254 0.91 KCNH2 (0.49) KCNH2CCR5
SCHEMBL4692674 0.90 KCNH2 (0.51) KCNH2CCR5
SCHEMBL4696713 0.90 KCNH2 (0.49) KCNH2CCR5
SCHEMBL4691753 0.90 KCNH2 (0.51) KCNH2CCR5
SCHEMBL4695092 0.90 CCR5 (0.51) KCNH2CCR5
SCHEMBL4745210 0.90 CCR5 (0.53) KCNH2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed