SCHEMBL4696266

SCHEMBL4696266

Cc1ccc(N(CCCN2CC3CN(C(=O)c4c(C)ccnc4C)CC3C2)C(=O)NC2CCN(C(=O)OCc3ccccc3)CC2)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 11/20 0.43
ENPP2 Q13822 5/20 0.41
CCL5 P13501 1/20 0.40
KCNH2 Q12809 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694200 0.89 CCR5 (0.44) CCR5KCNH2
SCHEMBL4696268 0.88 CCR5 (0.39) CCR5ENPP2KCNH2MEN1KMT2A
SCHEMBL4696397 0.87 CCR5 (0.48) CCR5CCL5KCNH2
SCHEMBL4691344 0.87 CCR5 (0.47) CCR5CCL5KCNH2
SCHEMBL4694951 0.83 CCR5 (0.48) CCR5CCL5
SCHEMBL4694411 0.82 CCR5 (0.45) CCR5CCL5KCNH2
Cyclopropane SCHEMBL4691469 0.81 CCR5 (0.48) CCR5CCL5KCNH2
Cyclopentane SCHEMBL4696746 0.81 CCR5 (0.48) CCR5CCL5KCNH2
Cyclohexane SCHEMBL4695443 0.81 CCR5 (0.48) CCR5CCL5KCNH2
SCHEMBL4691909 0.81 CCR5 (0.48) CCR5CCL5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1871762-A2 SUBTITUTED HETEROARYL CB1 ANTAGONISTS NEUROGEN CORPORATION (US) 2008-01-02 EP disclosed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed
WO-2006113704-A2 SUBTITUTED HETEROARYL CB1 ANTAGONISTS NEUROGEN CORPORATION (US) 2006-10-26 WO disclosed