SCHEMBL4696403

SCHEMBL4696403

Cc1ccc(N(CCCN2CC3=CN(C(=O)c4c(C)ccnc4C)CC3C2)C(=O)NCc2ccco2)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
UBE2M P61081 1/20 0.35
DCUN1D1 Q96GG9 1/20 0.35
CCR5 P51681 4/20 0.34
ALDH1A1 P00352 4/20 0.34
POLB P06746 2/20 0.34
KMT2A Q03164 1/20 0.34
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KCNH2 Q12809 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696925 0.89 CCR5 (0.40) CCR5ALDH1A1KCNH2
SCHEMBL4691464 0.88 CCR5 (0.37) CCR5KCNH2
SCHEMBL4694419 0.88 CCR5 (0.36) CCR5KCNH2
SCHEMBL4693620 0.87 CCR5 (0.44) CCR5KCNH2
SCHEMBL4694952 0.86 CCR5 (0.37) LMNAUBE2MDCUN1D1CCR5KCNH2
SCHEMBL4695967 0.86 CCR5 (0.36) CCR5ALDH1A1KCNH2
SCHEMBL4690669 0.86 CCR5 (0.45) CCR5KCNH2
SCHEMBL4696402 0.86 CCR5 (0.37) CCR5KCNH2
SCHEMBL4694980 0.86 CCR5 (0.42) L3MBTL1LMNAUBE2MDCUN1D1CCR5
SCHEMBL4694067 0.85 CCR5 (0.34) CCR5KMT2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed