SCHEMBL4696472

SCHEMBL4696472

O=C(O)N1CC2CN(C3Cc4ccccc4C3)CC2C1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 3/20 0.48
NPSR1 Q6W5P4 1/20 0.48
GRIN2B Q13224 2/20 0.42
BCHE P06276 6/20 0.42
ACHE P22303 1/20 0.42
S1PR5 Q9H228 1/20 0.40
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
LMNA P02545 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3019601 0.72 BPTF (0.48) ALDH1A1KDM4ENPSR1GRIN2BCHRNB2
SCHEMBL3316638 0.71 GRM7 (0.43) GRIN2BLMNAHRH3
SCHEMBL18498060 0.71 CHRNB2 (0.39) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL18498063 0.71 CHRNB2 (0.39) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL4694583 0.70 HRH3 (0.44) ALDH1A1KDM4ENPSR1LMNAHRH3
SCHEMBL5137807 0.69 CHRNB2 (0.44) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL7685605 0.68 GRIN2B (0.58) ALDH1A1GRIN2BS1PR5LMNA
SCHEMBL4692050 0.68 GRIN2B (0.58) ALDH1A1GRIN2BS1PR5LMNA
SCHEMBL4696479 0.67 BCHE (0.36) ALDH1A1KDM4ENPSR1GRIN2BBCHE
SCHEMBL14704615 0.67 GRIN2B (0.67) ALDH1A1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910374-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC SODIUM CHANNELS Vernalis (R&D) Limited (GB) 2008-04-16 EP disclosed
WO-2007007069-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC SODIUM CHANNELS VERNALIS (R & D) LIMITED (GB) 2007-01-18 WO disclosed