SCHEMBL4696504

SCHEMBL4696504

Nc1nc(NCc2ccc(F)cc2)nc(-c2cc(C3CC3)[nH]n2)c1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
NTRK1 P04629 3/20 0.46
MAPT P10636 5/20 0.44
KMT2A Q03164 2/20 0.44
HTT P42858 1/20 0.44
MEN1 O00255 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
MAPK1 P28482 2/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
PKM P14618 1/20 0.41
MGMT P16455 1/20 0.40
POLB P06746 1/20 0.40
PRKCQ Q04759 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3137390 0.86 HTT (0.46) CYP1A2CYP3A4CYP2C9CYP2C19NTRK1
SCHEMBL4696420 0.85 NTRK1 (0.51) CYP1A2CYP2C9CYP2C19NTRK1MKNK1
SCHEMBL4073888 0.84 NTRK1 (0.53) NTRK1MKNK1MKNK2
SCHEMBL3137650 0.82 HTT (0.48) CYP1A2CYP3A4CYP2C9CYP2C19NTRK1
SCHEMBL2571347 0.80 HTT (0.46) CYP1A2CYP3A4CYP2C9CYP2C19NTRK1
SCHEMBL3667400 0.79 NTRK1 (0.52) NTRK1PRKCQ
SCHEMBL3775237 0.79 NTRK1 (0.52) NTRK1PRKCQ
SCHEMBL2577693 0.79 PRKCQ (0.44) CYP1A2CYP3A4CYP2C9CYP2C19NTRK1
SCHEMBL3781156 0.78 JAK2 (0.50) NTRK1
SCHEMBL2569963 0.72 NTRK1 (0.48) CYP1A2CYP3A4CYP2C9CYP2C19NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1853588-B1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2008-06-18 EP disclosed