SCHEMBL3137650

SCHEMBL3137650

Nc1nc(NCc2ccc(F)cc2)c([N+](=O)[O-])c(-c2cc(C3CC3)[nH]n2)c1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.48
NTRK1 P04629 3/20 0.43
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAPT P10636 4/20 0.41
PRKCQ Q04759 1/20 0.41
LMNA P02545 2/20 0.40
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
KMT2A Q03164 2/20 0.38
MAPK1 P28482 1/20 0.38
HPGD P15428 1/20 0.38
MEN1 O00255 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPC1 O15118 1/20 0.37
MGMT P16455 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2571347 0.85 HTT (0.46) HTTNTRK1CYP1A2CYP3A4CYP2C9
SCHEMBL3137390 0.85 HTT (0.46) HTTNTRK1CYP1A2CYP3A4CYP2C9
SCHEMBL2577693 0.83 PRKCQ (0.44) HTTNTRK1CYP1A2CYP3A4CYP2C9
SCHEMBL4696504 0.82 CYP1A2 (0.49) HTTNTRK1CYP1A2CYP3A4CYP2C9
SCHEMBL3015513 0.80 NTRK1 (0.49) NTRK1
SCHEMBL3023274 0.78 JAK2 (0.47) NTRK1
SCHEMBL2566466 0.73 NTRK1 (0.48) NTRK1MKNK1MKNK2
SCHEMBL4696420 0.72 NTRK1 (0.51) NTRK1CYP1A2CYP2C9CYP2C19MKNK1
SCHEMBL4698162 0.72 NTRK1 (0.44) NTRK1SMN1; SMN2MAPK1MKNK1MKNK2
SCHEMBL2576261 0.71 NTRK1 (0.49) NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1853602-B1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2010-07-14 EP disclosed