SCHEMBL4698146

SCHEMBL4698146

NC1Cc2ccccc2-c2n[c]ncc21

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 4/20 0.36
NOS3 P29474 7/20 0.36
NOS2 P35228 5/20 0.34
HTR2A P28223 2/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
PLAU P00749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL148695 0.70 KDM4E (0.49) NOS3NOS2KDM4EALDH1A1POLB
SCHEMBL8006401 0.70 CYP3A4 (0.55) KDM4EALDH1A1
SCHEMBL4748664 0.69 HTR2A (0.58) ANPEPNOS3NOS2HTR2A
SCHEMBL467591 0.68 DRD4 (0.45) NOS3KDM4EALDH1A1POLB
SCHEMBL31373438 0.64
SCHEMBL2463276 0.64
SCHEMBL31373436 0.64
SCHEMBL20863915 0.64 HTR2A (0.35) ANPEPNOS3NOS2HTR2A
SCHEMBL18952772 0.64 MAPT (0.40) KDM4EALDH1A1POLB
SCHEMBL11185918 0.64 CDK8 (0.53) ANPEPNOS3NOS2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960382-A1 HETEROCYCLIC COMPOUNDS AS TYROSINE KINASE MODULATORS ChemBridge Research Laboratories, Inc. (US) 2008-08-27 EP disclosed
WO-2007056155-A1 HETEROCYCLIC COMPOUNDS AS TYROSINE KINASE MODULATORS CHEMBRIDGE RESEARCH LABORATORIES, INC. (US) 2007-05-18 WO disclosed