SCHEMBL4748664

SCHEMBL4748664

NC1Cc2ccccc2-c2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.58
ANPEP P15144 3/20 0.44
KDM1A O60341 4/20 0.42
NOS3 P29474 2/20 0.41
NOS2 P35228 2/20 0.41
HRH1 P35367 2/20 0.41
HTR2C P28335 1/20 0.41
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11185918 0.84 CDK8 (0.53) HTR2AANPEPKDM1ANOS3NOS2
SCHEMBL31373438 0.81
SCHEMBL31373436 0.81
SCHEMBL2463276 0.81
Hydrochloric Acid SCHEMBL19926846 0.79 KDM1A (0.57) HTR2AANPEPKDM1AHRH1HTR2C
Hydrochloric Acid SCHEMBL22635715 0.77 HTR2A (0.54) HTR2AANPEPKDM1AHRH1HTR2C
SCHEMBL24399522 0.77 S100A4 (0.52) HTR2AANPEPACHE
SCHEMBL20402534 0.77 PLAU (0.54) HTR2ANOS3NOS2ACHE
SCHEMBL14870745 0.76 HTR2A (0.55) HTR2ANOS3NOS2HRH1ACHE
SCHEMBL29439854 0.76 HTR2A (0.55) HTR2ANOS3NOS2HRH1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-52142054-A None JP disclosed
JP-52142054-A None JP disclosed
WO-2008123821-A1 4, 5-DIHYDRO-LH-IMIDAZOL-2-AMINE DERIVATIVES FOR USE IN THE TREATMENT OF RESPIRATORY, CARDIOVASCULAR, NEUROLOGICAL OR GASTROINTESTINAL DISORDERS ALBIREO AB (SE) 2008-10-16 WO disclosed
JP-S52142054-A 10-AMINO-9,10-DIHYROPHENANTHRENE DERIVATIVES AND THEIR PREPARATION RES INST FOR PROD DEV 1977-11-26 JP disclosed
JP-S52142054-A 10-AMINO-9,10-DIHYROPHENANTHRENE DERIVATIVES AND THEIR PREPARATION RES INST FOR PROD DEV 1977-11-26 JP disclosed