SCHEMBL4698291

SCHEMBL4698291

CC(C)(F)C(F)c1cccc(C2(N)CC2)c1.CC(C)(c1cccc(C2(N)CC2)c1)C(F)F

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.35
CTSD P07339 1/20 0.35
CYP3A4 P08684 1/20 0.35
KDM1A O60341 2/20 0.33
KCNN4 O15554 2/20 0.33
SLC6A4 P31645 2/20 0.33
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRL1 P41146 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4698709 0.89
SCHEMBL4698193 0.88 BACE1 (0.40) BACE1CTSDCYP3A4KDM1AKCNN4
SCHEMBL2351125 0.71 BACE1 (0.40) BACE1
SCHEMBL1420518 0.71 KDM1A (0.59) KDM1AKCNN4SLC6A4OPRL1SLC6A3
SCHEMBL4700710 0.70 KIF11 (0.36) CYP3A4
Hydrochloric Acid SCHEMBL3001569 0.70 KDM1A (0.57) KDM1AKCNN4SLC6A4OPRL1SLC6A3
SCHEMBL27426482 0.69 KDM1A (0.37) KDM1ASLC6A4
SCHEMBL2525890 0.68 KDM4E (0.39) CYP3A4
SCHEMBL2871341 0.68 KDM1A (0.41) BACE1KDM1AKCNN4SLC6A4
Hydrochloric Acid SCHEMBL3581155 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937638-A1 METHODS OF TREATING AMYLOIDOSIS USING ARYL-CYCLOPROPYL DERIVATIVE ASPARTYL PROTEASE INHIBITORS Elan Pharmaceuticals Inc. (US) 2008-07-02 EP disclosed
WO-2007047306-A1 METHODS OF TREATING AMYLOIDOSIS USING ARYL-CYCLOPROPYL DERIVATIVE ASPARTYL PROTEASE INHIBITORS ELAN PHARMACEUTICALS, INC. (US) 2007-04-26 WO disclosed