SCHEMBL4702249

SCHEMBL4702249

NC(=O)c1ccc(C2=NC(NC(=O)CCc3ccc(Cl)cc3Cl)C(=O)N(CCCN3CCCC3)c3ccccc32)cc1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.64
CCKBR P32239 8/20 0.46
OXTR P30559 7/20 0.46
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
CCKAR P32238 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4755895 0.99 KCNH2 (0.63) KCNH2CCKBROXTRPSEN1PSEN2
SCHEMBL4699817 0.94 KCNH2 (0.62) KCNH2CCKBROXTRPSEN1PSEN2
SCHEMBL4698132 0.91 KCNH2 (0.68) KCNH2CCKBROXTRPSEN1PSEN2
SCHEMBL4702302 0.88 KCNH2 (0.78) KCNH2CCKBROXTRPSEN1PSEN2
Hydrochloric Acid SCHEMBL4697415 0.87 KCNH2 (0.77) KCNH2CCKBROXTRPSEN1PSEN2
SCHEMBL4697333 0.85 KCNH2 (0.66) KCNH2CCKBRPSEN1PSEN2APH1B
SCHEMBL4697879 0.82 KCNH2 (0.62) KCNH2CCKBROXTRPSEN1PSEN2
SCHEMBL6076563 0.81 KCNH2 (0.54) KCNH2CCKBROXTRPSEN1PSEN2
SCHEMBL4699922 0.80 KCNH2 (0.59) KCNH2CCKBRPSEN1PSEN2APH1B
SCHEMBL7091166 0.78 KCNH2 (1.00) KCNH2CCKBROXTRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326849-B1 BENZODIAZEPINE DERIVATIVES AS INHIBITORS OF GAMMA SECRETASE MERCK SHARP & DOHME (GB) 2008-07-16 EP claimed