SCHEMBL4702302

SCHEMBL4702302

CN(C)CCCN1C(=O)C(NC(=O)CCc2ccc(Cl)cc2Cl)N=C(c2ccc(C(N)=O)cc2)c2ccccc21

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.78
OXTR P30559 6/20 0.48
CCKBR P32239 5/20 0.47
HDAC3 O15379 5/20 0.46
HDAC4 P56524 5/20 0.46
HDAC1 Q13547 5/20 0.46
HDAC7 Q8WUI4 5/20 0.46
HDAC2 Q92769 5/20 0.46
HDAC10 Q969S8 5/20 0.46
HDAC11 Q96DB2 5/20 0.46
HDAC8 Q9BY41 5/20 0.46
HDAC6 Q9UBN7 5/20 0.46
HDAC9 Q9UKV0 5/20 0.46
HDAC5 Q9UQL6 5/20 0.46
CCKAR P32238 1/20 0.45
PSEN1 P49768 1/20 0.45
PSEN2 P49810 1/20 0.45
APH1B Q8WW43 1/20 0.45
NCSTN Q92542 1/20 0.45
APH1A Q96BI3 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4697415 0.99 KCNH2 (0.77) KCNH2OXTRCCKBRHDAC3HDAC4
SCHEMBL4698132 0.91 KCNH2 (0.68) KCNH2OXTRCCKBRHDAC3HDAC4
SCHEMBL7091166 0.88 KCNH2 (1.00) KCNH2OXTRCCKBRHDAC3HDAC4
SCHEMBL4702249 0.88 KCNH2 (0.64) KCNH2OXTRCCKBRCCKARPSEN1
Hydrochloric Acid SCHEMBL4755895 0.87 KCNH2 (0.63) KCNH2OXTRCCKBRCCKARPSEN1
SCHEMBL4697333 0.87 KCNH2 (0.66) KCNH2CCKBRHDAC3HDAC4HDAC1
SCHEMBL4699817 0.86 KCNH2 (0.62) KCNH2OXTRCCKBRCCKARPSEN1
Hydrochloric Acid SCHEMBL6003884 0.86 KCNH2 (0.60) KCNH2OXTRCCKBRCCKARPSEN1
SCHEMBL4697879 0.84 KCNH2 (0.62) KCNH2OXTRCCKBRCCKARPSEN1
SCHEMBL4699922 0.82 KCNH2 (0.59) KCNH2CCKBRHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326849-B1 BENZODIAZEPINE DERIVATIVES AS INHIBITORS OF GAMMA SECRETASE MERCK SHARP & DOHME (GB) 2008-07-16 EP claimed