SCHEMBL470298

SCHEMBL470298

Cc1[nH]nc(C2CC=CC=C2Cl)c1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.36
TTR P02766 1/20 0.31
DAO P14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL470472 0.73 NOTUM (0.42)
SCHEMBL902697 0.72 GAA (0.32)
SCHEMBL10081881 0.70 KDM4E (0.40)
SCHEMBL21834224 0.69 HCAR2 (0.40) HCAR2DAO
SCHEMBL470311 0.64 PDE4D (0.30)
SCHEMBL22637228 0.63 FABP4 (0.34) HCAR2DAO
SCHEMBL1663754 0.60 PDE4D (0.59) HCAR2TTRDAO
SCHEMBL27575758 0.59 HCAR2 (0.61) HCAR2DAO
SCHEMBL903102 0.59
SCHEMBL22637832 0.58 HCAR2 (0.41) HCAR2DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044531-A1 NOVEL PIPERAZINE ANALOGS WITH SUBSTITUTED HETEROARYL GROUPS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-04-05 WO disclosed
WO-2012033736-A1 NOVEL PIPERAZINE ANALOGS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-15 WO disclosed