SCHEMBL4704258

SCHEMBL4704258

CCCCN[C@H](C(=O)O)[C@@H](C)CC

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.46
MAPK1 P28482 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
PLA2G2A P14555 1/20 0.41
PLA2G5 P39877 1/20 0.41
CA2 P00918 2/20 0.41
ALOX15 P16050 1/20 0.41
FPR2 P25090 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
MME P08473 1/20 0.38
ACE P12821 1/20 0.38
CPA1 P15085 1/20 0.38
ACE2 Q9BYF1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4704256 1.00 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2MAPK1L3MBTL1PLA2G2A
SCHEMBL9828860 0.94 SMN1; SMN2 (0.53) ALDH1A1SMN1; SMN2MAPK1L3MBTL1PLA2G2A
Water SCHEMBL27944924 0.92 SMN1; SMN2 (0.51) ALDH1A1SMN1; SMN2MAPK1L3MBTL1PLA2G2A
SCHEMBL17939720 0.92 SMN1; SMN2 (0.51) ALDH1A1SMN1; SMN2MAPK1L3MBTL1PLA2G2A
SCHEMBL11796686 0.92 SMN1; SMN2 (0.51) ALDH1A1SMN1; SMN2MAPK1L3MBTL1PLA2G2A
SCHEMBL26122722 0.92 SMN1; SMN2 (0.51) ALDH1A1SMN1; SMN2MAPK1L3MBTL1PLA2G2A
SCHEMBL11800511 0.92 SMN1; SMN2 (0.51) ALDH1A1SMN1; SMN2MAPK1L3MBTL1PLA2G2A
SCHEMBL27905915 0.92 SMN1; SMN2 (0.51) ALDH1A1SMN1; SMN2MAPK1L3MBTL1PLA2G2A
SCHEMBL28031785 0.91 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2MAPK1L3MBTL1PLA2G2A
SCHEMBL28032316 0.91 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2MAPK1L3MBTL1PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599471-B1 HYDROXYMETHYL SUBSTITUTED DIHYDROISOXAZOLE DERIVATIVES USEFUL AS ANTIBIOTIC AGENTS ASTRAZENECA AB (SE) 2008-05-28 EP disclosed
EP-0157963-B1 6H-DIBENZ (B,E)(1,4)OXATHIEPIN COMPOUNDS MERCK & CO. INC. (US) 1989-06-21 EP disclosed
US-4778897-A 6H-dibenz[b,e][1,4]oxathiepin compounds MERCK & CO., INC. (US) 1988-10-18 US disclosed
US-4699917-A Anti-asthmatic tetrazolyl 6H-dibenz-[B,E]-[1,4]-oxathiepin derivatives, compositions, and method of use therefor MERCK & CO., INC. (US) 1987-10-13 US disclosed
EP-0069810-B1 NOVEL DIBENZOXEPINS, THEIR PREPARATION, COMPOSITIONS CONTAINING THEM AND THE USE OF DIBENZOXEPINS IN THE TREATMENT OF ALLERGIC CONDITIONS MERCK & CO. INC. (US) 1986-12-03 EP disclosed
US-4582842-A Anti-asthmatic 6H-dibenz-[b,e] [1,4]oxathiepin derivatives, compositions, and method of use therefor MERCK & CO., INC. (US) 1986-04-15 US disclosed
EP-0157963-A1 6H-dibenz (b,e)(1,4)oxathiepin compounds MERCK & CO. INC. (US) 1985-10-16 EP disclosed
US-4536507-A ANTIASTHMA AGENTS MERCK & CO., INC. (US) 1985-08-20 US disclosed
US-4394515-A 10,11-Dihydro-11-oxodibenzo[b,f]thiepin compounds MERCK & CO., INC. (US) 1983-07-19 US disclosed
EP-0069810-A1 Novel dibenzoxepins, their preparation, compositions containing them and the use of dibenzoxepins in the treatment of allergic conditions MERCK & CO. INC. (US) 1983-01-19 EP disclosed
EP-0000978-B1 7-AND 8-SUBSTITUTED -10,11-DIHYDRO-11-OXODIBENZO (B,F) THIEPIN DERIVATIVES, THEIR PRODUCTION AND THEIR PARMACEUTICAL COMPOSITIONS MERCK & CO. INC. (US) 1982-09-15 EP disclosed
US-4282365-A Dibenz[b,e]oxepin compounds MERCK & CO., INC. (US) 1981-08-04 US disclosed
US-4263207-A ANTIALLERGENS MERCK & CO., INC. (US) 1981-04-21 US disclosed
EP-0011067-A1 Prostaglandin antagonists, their production and their pharmaceutical compositions MERCK & CO. INC. (US) 1980-05-28 EP disclosed
EP-0000978-A1 7-and 8-substituted -10,11-dihydro-11-oxodibenzo (b,f) thiepin derivatives, their production and their parmaceutical compositions MERCK & CO. INC. (US) 1979-03-07 EP disclosed