SCHEMBL470435

SCHEMBL470435

O=C(O)c1cnc(C[C@@H]2CCOC2)c(-c2ccc(Cl)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 12/20 0.44
XDH P47989 1/20 0.41
MAP4K4 O95819 2/20 0.40
CNR2 P34972 2/20 0.39
MAPK1 P28482 1/20 0.39
GPR119 Q8TDV5 1/20 0.38
BRS3 P32247 1/20 0.37
GRM4 Q14833 1/20 0.36
KDM4C Q9H3R0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16938615 0.89 CNR1 (0.54) CNR1XDHMAP4K4CNR2MAPK1
SCHEMBL410543 0.83 CNR1 (0.55) CNR1XDHCNR2GRM4
SCHEMBL412004 0.76 CNR1 (0.52) CNR1CNR2
SCHEMBL441630 0.76 CNR1 (0.52) CNR1CNR2
SCHEMBL442354 0.71 CNR1 (0.67) CNR1CNR2
SCHEMBL27973515 0.70 CHEK1 (0.54)
SCHEMBL442533 0.70 MAP4K4 (0.55) CNR1MAP4K4
SCHEMBL2702006 0.68 MARS1 (0.46) CNR1MAP4K4
SCHEMBL411076 0.67 CNR1 (0.67) CNR1MAP4K4CNR2
SCHEMBL5355700 0.66 CNR1 (0.67) CNR1MAP4K4CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012032018-A1 HETEROARYLMETHYL AMIDES F. HOFFMANN-LA ROCHE AG (CH) 2012-03-15 WO disclosed