SCHEMBL4707138

SCHEMBL4707138

O=C(NCc1ccccc1Cl)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1cnccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C19 P33261 2/20 0.47
TP53 P04637 3/20 0.46
MAPT P10636 5/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
CNR2 P34972 1/20 0.41
ROCK2 O75116 1/20 0.41
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.40
TSHR P16473 1/20 0.40
THRB P10828 2/20 0.40
POLB P06746 2/20 0.40
CACNA1G O43497 2/20 0.40
CACNA1H O95180 2/20 0.40
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4706658 0.88 IDH1 (0.62) IDH1CYP1A2CYP3A4CYP2C19TP53
SCHEMBL4706587 0.86 IDH1 (0.52) IDH1CYP1A2CYP3A4CYP2C19TP53
SCHEMBL4705917 0.85 IDH1 (0.50) IDH1CYP1A2CYP3A4CYP2C19TP53
SCHEMBL4706712 0.83 TP53 (0.52) IDH1CYP1A2CYP3A4CYP2C19TP53
SCHEMBL4637887 0.80 USP2 (0.36) IDH1CYP3A4KMT2AMEN1TSHR
SCHEMBL4707944 0.80 IDH1 (0.48) IDH1TP53ALDH1A1GAATSHR
SCHEMBL4705941 0.79 TP53 (0.50) CYP1A2CYP3A4CYP2C19TP53MAPT
SCHEMBL4637963 0.79 USP2 (0.45) CYP1A2CYP3A4CYP2C19KMT2AMEN1
SCHEMBL4638494 0.78 USP2 (0.42) CYP1A2CYP3A4TP53MAPTKMT2A
SCHEMBL4707117 0.78 TACR1 (0.45) CYP1A2CYP3A4CYP2C19TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed