SCHEMBL4707944

SCHEMBL4707944

O=C(NCc1cccc(Cl)c1Cl)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.48
CACNA1G O43497 2/20 0.46
CACNA1H O95180 2/20 0.46
TP53 P04637 1/20 0.44
TACR1 P25103 7/20 0.43
CCR1 P32246 1/20 0.42
ALDH1A1 P00352 2/20 0.42
GAA P10253 1/20 0.42
PTGER4 P35408 1/20 0.41
CYP19A1 P11511 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705917 0.94 IDH1 (0.50) IDH1CACNA1GCACNA1HTP53TACR1
SCHEMBL4706587 0.88 IDH1 (0.52) IDH1CACNA1GCACNA1HTP53ALDH1A1
SCHEMBL4707843 0.87 EPHX2 (0.48) IDH1CACNA1GCACNA1HTACR1ALDH1A1
SCHEMBL4708123 0.87 TP53 (0.49) IDH1CACNA1GCACNA1HTP53TACR1
SCHEMBL4706714 0.86 TACR1 (0.48) IDH1CACNA1GCACNA1HTACR1ALDH1A1
SCHEMBL4706969 0.86 CACNA1G (0.49) IDH1CACNA1GCACNA1HTP53TACR1
SCHEMBL4707735 0.86 TACR1 (0.52) IDH1TP53TACR1ALDH1A1GAA
SCHEMBL4706658 0.85 IDH1 (0.62) IDH1CACNA1GCACNA1HTP53TACR1
SCHEMBL4707851 0.83 GRM2 (0.40) IDH1CACNA1GCACNA1HTP53TACR1
SCHEMBL4706967 0.83 POLB (0.50) IDH1TACR1ALDH1A1GAAPTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed