SCHEMBL4707159

SCHEMBL4707159

COc1cc(C(=O)[C@@H]2C(=O)c3cc(-c4cccc(C(=O)O)c4)ccc3OC23CCNCC3)cc2c(C3CC3)nccc12

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.34
PDE4B Q07343 2/20 0.34
PDE4A P27815 1/20 0.34
PDE4C Q08493 1/20 0.34
ACACB O00763 2/20 0.32
ACACA Q13085 2/20 0.32
HSD17B13 Q7Z5P4 1/20 0.32
NR1H4 Q96RI1 1/20 0.32
IMPDH2 P12268 1/20 0.31
FYN P06241 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4710321 0.94 PDE4D (0.35) PDE4DNR1H4
SCHEMBL4708956 0.87 ACACB (0.35) ACACBACACA
SCHEMBL4710166 0.87 ACACB (0.35) ACACBACACA
SCHEMBL4708849 0.85
SCHEMBL3859694 0.81 ACACB (0.40) PDE4DPDE4BPDE4APDE4CACACB
SCHEMBL4709624 0.80 ACACB (0.31) ACACBACACA
SCHEMBL4758667 0.79
SCHEMBL4757588 0.78
SCHEMBL4759844 0.78
SCHEMBL4276308 0.78 ACACB (0.43) PDE4DPDE4BPDE4APDE4CACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910375-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS Merck & Co., Inc. (US) 2008-04-16 EP disclosed
WO-2007011809-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS MERCK & CO., INC. (US) 2007-01-25 WO disclosed