SCHEMBL4707652

SCHEMBL4707652

FC(F)(F)c1cc(Cn2nnc(-c3cn[nH]c3Cc3ccccc3Cl)c2-c2ccccc2)cc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 9/20 0.44
MAP4K4 O95819 5/20 0.44
PRKACA P17612 5/20 0.44
CDK2 P24941 5/20 0.44
GSK3B P49841 5/20 0.44
CLK4 Q9HAZ1 4/20 0.44
MKNK2 Q9HBH9 4/20 0.44
PIM1 P11309 3/20 0.44
HIPK2 Q9H2X6 3/20 0.44
DAPK3 O43293 4/20 0.39
ROCK2 O75116 4/20 0.39
PRKD3 O94806 4/20 0.39
CLK2 P49760 4/20 0.39
PRKX P51817 4/20 0.39
JAK3 P52333 4/20 0.39
CDK5 Q00535 4/20 0.39
MAP4K2 Q12851 4/20 0.39
CAMK2D Q13557 4/20 0.39
DYRK1A Q13627 4/20 0.39
PKN2 Q16513 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708541 0.88 CDC7 (0.41) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4706683 0.84 CDC7 (0.38) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL14279260 0.80 CDC7 (0.42) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4707969 0.80 CDC7 (0.42) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4706420 0.79 IDO1 (0.44) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4705965 0.78 POLB (0.48) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4707886 0.77 GRM2 (0.36) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4705832 0.76 GRM2 (0.38) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4707214 0.76 CDC7 (0.39) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4706369 0.76 P2RX7 (0.45) CDC7MAP4K4PRKACACDK2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed