SCHEMBL4708335

SCHEMBL4708335

Cc1cccc(NC(=O)C2CNCCN2c2nc(N)nc3ccc(-c4ccccc4)nc23)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.44
POLB P06746 1/20 0.44
ALDH1A1 P00352 3/20 0.42
PI4KB Q9UBF8 1/20 0.40
MKNK2 Q9HBH9 2/20 0.38
TSHR P16473 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GAA P10253 1/20 0.37
USP2 O75604 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
ALOX12 P18054 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
KCNH2 Q12809 1/20 0.36
CCNC P24863 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4118504 0.94 PI4KB (0.39) MAPTPOLBALDH1A1PI4KBTSHR
SCHEMBL4107810 0.92 POLB (0.39) MAPTPOLBALDH1A1PI4KBMKNK2
SCHEMBL4108347 0.92 MKNK1 (0.38) MAPTPOLBALDH1A1PI4KBMKNK2
SCHEMBL4116800 0.91 PI4KB (0.40) MAPTPOLBALDH1A1PI4KBTSHR
SCHEMBL4102550 0.91 POLB (0.38) MAPTPOLBALDH1A1PI4KBTSHR
SCHEMBL4101466 0.91 MKNK2 (0.39) MAPTPOLBALDH1A1PI4KBMKNK2
SCHEMBL4108372 0.89 ALDH1A1 (0.39) MAPTPOLBALDH1A1PI4KBTSHR
SCHEMBL4121021 0.89 ALDH1A1 (0.38) MAPTPOLBALDH1A1PI4KBTSHR
SCHEMBL4521469 0.89 PDE4A (0.51) MAPTPOLBALDH1A1PI4KBUSP2
SCHEMBL3922088 0.88 ALDH1A1 (0.40) MAPTPOLBALDH1A1PI4KBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899332-A1 PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING HEPATITIS C. GILEAD SCIENCES, INC. (US) 2008-03-19 EP disclosed
WO-2006135993-A1 PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS USEFUL FOR TREATING HEPATITIS C. GILEAD SCIENCES, INC. (US) 2006-12-28 WO disclosed