SCHEMBL4709130

SCHEMBL4709130

COC(=O)c1ccc(C=Cc2cc3c(cc2CCO)C(C)(C)CCC3(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RARB P10826 8/20 0.52
RARG P13631 8/20 0.52
RARA P10276 7/20 0.52
CYP3A4 P08684 3/20 0.47
CYP26A1 O43174 3/20 0.44
PTPN1 P18031 1/20 0.44
VDR P11473 4/20 0.43
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
NPC1 O15118 2/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
CYP4F2 P78329 1/20 0.40
CYP4A11 Q02928 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4669351 1.00 RARB (0.52) RARBRARGRARACYP3A4CYP26A1
SCHEMBL4666486 0.94 RARB (0.50) RARBRARGRARACYP3A4CYP26A1
SCHEMBL4666454 0.94 RARB (0.50) RARBRARGRARACYP3A4CYP26A1
SCHEMBL6909571 0.91 RARB (0.52) RARBRARGRARACYP3A4CYP26A1
SCHEMBL10842924 0.90 RARB (0.55) RARBRARGRARACYP3A4CYP26A1
SCHEMBL10842927 0.90 RARB (0.55) RARBRARGRARACYP3A4CYP26A1
SCHEMBL10843882 0.89 RARA (0.50) RARBRARGRARACYP3A4CYP26A1
SCHEMBL10843886 0.89 RARA (0.50) RARBRARGRARACYP3A4CYP26A1
SCHEMBL10847379 0.88 RARB (0.49) RARBRARGRARACYP3A4CYP26A1
SCHEMBL10847377 0.88 RARB (0.49) RARBRARGRARACYP3A4CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1935869-A1 Retinoids for the treatment of emphysema F. HOFFMANN-LA ROCHE AG (CH) 2008-06-25 EP disclosed
EP-1324970-A2 RETINOIDS FOR THE TREATMENT OF EMPHYSEMA F. HOFFMANN-LA ROCHE AG (CH) 2003-07-09 EP disclosed
WO-2002028810-A2 RETINOIDS FOR THE TREATMENT OF EMPHYSEMA F. HOFFMANN-LA ROCHE AG (CH) 2002-04-11 WO disclosed