SCHEMBL4710076

SCHEMBL4710076

COc1cc(Oc2ccnc3ccc(F)cc23)ccc1CC(=O)Nc1cn[nH]c1

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 19/20 0.72
CSF1R P07333 16/20 0.72
KDR P35968 15/20 0.72
FLT3 P36888 6/20 0.57
PDGFRA P16234 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5009418 0.88 KDR (0.56) PDGFRBCSF1RKDRFLT3PDGFRA
SCHEMBL4708414 0.87 PDGFRB (0.73) PDGFRBCSF1RKDRFLT3PDGFRA
SCHEMBL2174909 0.85 PDGFRB (0.82) PDGFRBCSF1RKDRFLT3PDGFRA
SCHEMBL2173586 0.84 PDGFRB (1.00) PDGFRBCSF1RKDRFLT3PDGFRA
SCHEMBL2174490 0.82 PDGFRB (0.69) PDGFRBCSF1RKDRFLT3PDGFRA
SCHEMBL2173264 0.82 PDGFRB (0.78) PDGFRBCSF1RKDRFLT3PDGFRA
SCHEMBL2176270 0.82 PDGFRB (0.66) PDGFRBCSF1RKDRFLT3PDGFRA
SCHEMBL2173476 0.80 PDGFRB (0.67) PDGFRBCSF1RKDRFLT3PDGFRA
SCHEMBL2177245 0.80 PDGFRB (1.00) PDGFRBCSF1RKDRFLT3PDGFRA
SCHEMBL22089482 0.78 PDGFRA (0.71) PDGFRBCSF1RKDRFLT3PDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1994025-A1 QUINOLINE DERIVATIVES AstraZeneca AB (SE) 2008-11-26 EP claimed
WO-2007099326-A1 QUINOLINE DERIVATIVES ASTRAZENECA AB (SE) 2007-09-07 WO claimed
EP-1994025-A1 QUINOLINE DERIVATIVES AstraZeneca AB (SE) 2008-11-26 EP disclosed
WO-2007099326-A1 QUINOLINE DERIVATIVES ASTRAZENECA AB (SE) 2007-09-07 WO disclosed