SCHEMBL4710102

SCHEMBL4710102

COc1cc(OC)c2cnc(-c3cc(C)c(OCC(C)(C)O)c(C)c3)cc2c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 10/20 0.40
IDO1 P14902 8/20 0.40
NPC1 O15118 5/20 0.40
RAB9A P51151 5/20 0.40
CASP3 P42574 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
BRD4 O60885 3/20 0.35
CYP1A1 P04798 1/20 0.34
CYP1B1 Q16678 1/20 0.34
HDAC1 Q13547 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL348838 0.81 TDO2 (0.52) TDO2IDO1NPC1RAB9ACASP3
SCHEMBL347960 0.79 IDO1 (0.46) TDO2IDO1NPC1RAB9ABRD4
SCHEMBL28288872 0.77 TDO2 (0.53) TDO2IDO1NPC1RAB9ACASP3
SCHEMBL348270 0.74 SYK (0.51) NPC1BRD4MEN1KMT2A
SCHEMBL348727 0.72 TDO2 (0.60) TDO2IDO1NPC1RAB9ACASP3
SCHEMBL145706 0.71 BRD4 (0.46) BRD4HDAC1
SCHEMBL30434678 0.71 BRD4 (0.46) BRD4HDAC1
SCHEMBL28288947 0.70 TDO2 (0.64) TDO2IDO1NPC1RAB9ACASP3
SCHEMBL28290268 0.69 TDO2 (0.65) TDO2IDO1NPC1RAB9ACASP3
SCHEMBL22635791 0.69 IDO1 (0.33) TDO2IDO1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1909788-A2 PHARMACEUTICAL COMPOSITIONS FOR THE PREVENTION AND TREATMENT OF COMPLEX DISEASES AND THEIR DELIVERY BY INSERTABLE MEDICAL DEVICES RESVERLOGIX CORP. (CA) 2008-04-16 EP claimed
WO-2007016525-A2 PHARMACEUTICAL COMPOSITIONS FOR THE PREVENTION AND TREATMENT OF COMPLEX DISEASES AND THEIR DELIVERY BY INSERTABLE MEDICAL DEVICES RESVERLOGIX CORP. (CA) 2007-02-08 WO claimed