SCHEMBL4710643

SCHEMBL4710643

Cc1cc(F)ccc1[C@H]1C[C@@H](N2CCN3C(=O)CCC3C2)CCN1OC(=O)N(C)Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.64
PTAFR P25105 1/20 0.64
SIGMAR1 Q99720 1/20 0.64
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2484832 0.88 TACR1 (0.77) TACR1PTAFRSIGMAR1CYP3A4
SCHEMBL3245145 0.87 TACR1 (0.66) TACR1SIGMAR1CYP3A4
SCHEMBL4707782 0.87 TACR1 (0.80) TACR1PTAFRSIGMAR1CYP3A4
SCHEMBL4712181 0.87 TACR1 (0.80) TACR1PTAFRSIGMAR1CYP3A4
Hydrochloric Acid SCHEMBL4709532 0.86 TACR1 (0.79) TACR1PTAFRSIGMAR1CYP3A4
SCHEMBL3244347 0.86 TACR1 (0.77) TACR1SIGMAR1CYP3A4
SCHEMBL3247986 0.86 TACR1 (0.77) TACR1SIGMAR1CYP3A4
SCHEMBL25277637 0.83 TACR1 (0.76) TACR1PTAFRSIGMAR1CYP3A4
SCHEMBL4709667 0.82 TACR1 (0.54) TACR1PTAFRSIGMAR1
SCHEMBL2483424 0.80 TACR1 (0.60) TACR1PTAFRSIGMAR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1666465-B1 Composition comprising a tachykinin receptor antagonist and a selective serotonin reuptake inhibitor GLAXO GROUP LTD (GB) 2008-05-07 EP claimed