SCHEMBL3245145

SCHEMBL3245145

Cc1cc(F)ccc1[C@H]1C[C@H](N2CCN(C)CC2)CCN1OC(=O)N(C)Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.66

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.66
CYP3A4 P08684 2/20 0.51
SIGMAR1 Q99720 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244347 0.92 TACR1 (0.77) TACR1CYP3A4SIGMAR1
SCHEMBL3247986 0.92 TACR1 (0.77) TACR1CYP3A4SIGMAR1
SCHEMBL4710643 0.87 TACR1 (0.64) TACR1CYP3A4SIGMAR1
SCHEMBL3248437 0.85 TACR1 (0.68) TACR1CYP3A4SIGMAR1
SCHEMBL6248151 0.81 TACR1 (0.66) TACR1
SCHEMBL4029704 0.81 TACR1 (0.73) TACR1
SCHEMBL3246935 0.81 TACR1 (0.80) TACR1CYP3A4SIGMAR1
SCHEMBL13627551 0.80 TACR1 (1.00) TACR1CYP3A4SIGMAR1
SCHEMBL13627555 0.80 TACR1 (1.00) TACR1CYP3A4SIGMAR1
SCHEMBL13627550 0.80 TACR1 (1.00) TACR1CYP3A4SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1921064-B1 Pharmaceutical composition GLAXO GROUP LTD (GB) 2010-05-19 EP claimed
EP-1524266-B1 Pharmaceutical composition GLAXO GROUP LTD (GB) 2007-02-28 EP claimed
EP-1326832-B1 CHEMICAL COMPOUNDS GLAXO GROUP LTD (GB) 2004-10-06 EP claimed
EP-1979349-B1 ANTI-VIRAL COMPOUNDS ABBOTT LAB (US) 2010-07-28 EP disclosed