SCHEMBL4710936

SCHEMBL4710936

Cc1ccc(OCCCN(C)C)c(C=Cc2ccccc2)n1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 2/20 0.45
BCHE P06276 5/20 0.44
ACHE P22303 5/20 0.44
HRH1 P35367 1/20 0.43
HRH3 Q9Y5N1 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
LSS P48449 1/20 0.40
TOP2A P11388 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4710935 1.00 HTR1B (0.45) HTR1BBCHEACHEHRH1HRH3
Hydrochloric Acid SCHEMBL4713327 0.99 HTR1B (0.44) HTR1BBCHEACHEHRH1HRH3
Hydrochloric Acid SCHEMBL4713323 0.99 HTR1B (0.44) HTR1BBCHEACHEHRH1HRH3
SCHEMBL4713204 0.88 HRH3 (0.44) HTR1BHRH3CYP1A2CYP2D6CYP2C19
SCHEMBL4713201 0.88 HRH3 (0.44) HTR1BHRH3CYP1A2CYP2D6CYP2C19
SCHEMBL27541419 0.87 ALDH1A1 (0.43) HTR1BBCHEACHEHRH1CYP2D6
Hydrochloric Acid SCHEMBL4711111 0.86 HRH3 (0.43) HRH3CYP1A2CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL4711116 0.86 HRH3 (0.43) HRH3CYP1A2CYP2D6CYP2C19
SCHEMBL4711191 0.86 CYP1A2 (0.46) HTR1BBCHEACHEHRH1CYP1A2
SCHEMBL4711192 0.86 CYP1A2 (0.46) HTR1BBCHEACHEHRH1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998459-B1 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 2008-04-23 EP claimed
EP-0998459-A2 PYRIDINE DERIVATIVES Novartis AG (CH) 2000-05-10 EP claimed
WO-1999002497-A2 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 1999-01-21 WO claimed