SCHEMBL4711098

SCHEMBL4711098

Cc1ccc(NC(=O)N[C@@H](C)c2cccc(CN3CCN([S+]([O-])N(C)C)CC3)c2)cn1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPK1 P28482 1/20 0.40
ACKR3 P25106 4/20 0.39
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
NAMPT P43490 4/20 0.38
CYP2C9 P11712 2/20 0.37
HTR1A P08908 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
WNT1 P04628 1/20 0.36
CLK2 P49760 1/20 0.36
CLK3 P49761 1/20 0.36
DYRK1A Q13627 1/20 0.36
OPRD1 P41143 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4710480 0.85 MEN1 (0.46) MEN1KMT2AMAPK1ACKR3ROCK2
SCHEMBL3736252 0.84 NAMPT (0.42) MEN1KMT2AMAPK1ACKR3ROCK2
SCHEMBL3742162 0.84 NAMPT (0.42) MEN1KMT2AMAPK1ACKR3ROCK2
Hydrochloric Acid SCHEMBL3739080 0.83 MAPK1 (0.43) MEN1KMT2AMAPK1ACKR3ROCK2
Hydrochloric Acid SCHEMBL3739075 0.83 MAPK1 (0.43) MEN1KMT2AMAPK1ACKR3ROCK2
SCHEMBL3731076 0.80 CCNK (0.42) MEN1KMT2AMAPK1ACKR3ROCK2
SCHEMBL3731078 0.80 CCNK (0.42) MEN1KMT2AMAPK1ACKR3ROCK2
SCHEMBL10315552 0.71 ACKR3 (0.57) ACKR3HTR1AHTR1DHTR1BNPSR1
SCHEMBL398679 0.71 ACKR3 (0.51) ACKR3CYP2C9HTR1AHTR1DHTR1B
SCHEMBL401714 0.70 ACKR3 (0.49) ACKR3HTR1AHTR1DHTR1BNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959963-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS Cytokinetics, Inc. (US) 2008-08-27 EP claimed
WO-2007089336-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2007-08-09 WO claimed