SCHEMBL4714048

SCHEMBL4714048

O=C(NC1CC1)NC1C=CC=CC1(Cl)Oc1ncnc2[nH]c(-c3ccc(OC[C@H](O)CN4CCCC4)cc3)cc12

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.37
MAPK1 P28482 1/20 0.37
ABCB1 P08183 5/20 0.36
ATM Q13315 1/20 0.36
CYP2D6 P10635 2/20 0.36
POLB P06746 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
TBK1 Q9UHD2 3/20 0.36
CYP2C19 P33261 1/20 0.35
ALOX15 P16050 1/20 0.35
RECQL P46063 1/20 0.35
ESR2 Q92731 1/20 0.35
SCN1A P35498 1/20 0.35
SCN5A Q14524 1/20 0.35
SCN9A Q15858 1/20 0.35
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14423908 0.81 KDR (0.44) KITMAPK1
SCHEMBL1896037 0.81 KDR (0.44) KITMAPK1
SCHEMBL1896040 0.81 KDR (0.44) KITMAPK1
SCHEMBL1895332 0.80 KDR (0.53)
SCHEMBL1891779 0.80 KDR (0.53)
SCHEMBL1892317 0.68 KDR (0.61) TBK1
SCHEMBL1895844 0.68 KDR (0.54) KIT
SCHEMBL12411681 0.67 FLT1 (0.66)
SCHEMBL1890518 0.67 KDR (0.38) KIT
SCHEMBL1890519 0.67 KDR (0.38) KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506962-B1 Nitrogen-containing aromatic heterocycles EISAI R&D MAN CO LTD (JP) 2008-07-02 EP disclosed