SCHEMBL4715260

SCHEMBL4715260

CCc1c(Oc2cc(Cl)cc(C#N)c2)c(CBr)nn1C(C)=O

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.51
CYP3A4 P08684 2/20 0.37
MAPT P10636 1/20 0.35
PGR P06401 6/20 0.34
EPAS1 Q99814 3/20 0.33
VEGFA P15692 2/20 0.33
ARNT P27540 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
RORC P51449 1/20 0.32
ADRA1D P25100 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL508819 0.88 KCNH2 (0.47) KCNH2CYP3A4MAPTEPAS1VEGFA
SCHEMBL509554 0.85 KCNH2 (0.52) KCNH2PGRPTGDR2RORC
SCHEMBL14304003 0.84 KCNH2 (0.49) KCNH2PGRRORC
SCHEMBL10251125 0.78 KCNH2 (0.42) KCNH2PGRPTGDR2
SCHEMBL14540679 0.77 KCNH2 (0.47) KCNH2CYP3A4MAPTEPAS1VEGFA
SCHEMBL508737 0.76 KCNH2 (0.42) KCNH2PGRRORC
SCHEMBL508806 0.76 MAPT (0.41) KCNH2MAPTPTGDR2
SCHEMBL508808 0.75 CYP3A4 (0.38) KCNH2CYP3A4EPAS1VEGFA
SCHEMBL4720561 0.75 KCNH2 (0.38) KCNH2CYP3A4PGRRORC
SCHEMBL508348 0.75 ENPP3 (0.45) KCNH2CYP3A4MAPTEPAS1VEGFA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551828-B1 PYRAZOLE DERIVATIVES PFIZER LTD (GB) 2008-01-23 EP disclosed