SCHEMBL4716351

SCHEMBL4716351

Nc1nc(Nc2ccccc2)ncc1/C=C/C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.47
AURKA O14965 5/20 0.47
GSK3A P49840 3/20 0.47
HDAC6 Q9UBN7 1/20 0.44
JAK2 O60674 2/20 0.44
AURKB Q96GD4 2/20 0.44
BCL6 P41182 1/20 0.44
ITK Q08881 2/20 0.43
EGFR P00533 2/20 0.43
RHOA P61586 1/20 0.43
MAPK8 P45983 3/20 0.42
IGF1R P08069 2/20 0.42
MAPK1 P28482 2/20 0.42
RAB9A P51151 2/20 0.42
SYK P43405 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
PKM P14618 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4716354 1.00 GSK3B (0.47) GSK3BAURKAGSK3AHDAC6JAK2
SCHEMBL4714877 0.83 EGFR (0.50) AURKAITKEGFRRAB9ANPC1
SCHEMBL4714874 0.83 EGFR (0.50) AURKAITKEGFRRAB9ANPC1
SCHEMBL4714696 0.81 BCL6 (0.50) GSK3BAURKAGSK3AHDAC6JAK2
SCHEMBL4715101 0.78 EGFR (0.47) GSK3BAURKAGSK3AJAK2AURKB
SCHEMBL4715103 0.78 EGFR (0.47) GSK3BAURKAGSK3AJAK2AURKB
SCHEMBL20953571 0.74 RAB9A (0.59) GSK3BAURKAGSK3AJAK2AURKB
SCHEMBL25345948 0.73 PLAU (0.44) HDAC6RAB9ATSHRNFKB1CLK4
SCHEMBL10187855 0.71 BCL6 (0.53) GSK3BAURKAGSK3AJAK2AURKB
SCHEMBL28223543 0.71 JAK2 (0.62) GSK3BAURKAGSK3AJAK2AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0964864-B1 PYRIDO 2,3-D PYRIMIDINES AND 4-AMINOPYRIMIDINES AS INHIBITORS OF CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2008-04-09 EP claimed