SCHEMBL4716562

SCHEMBL4716562

COc1cc(NCC(=O)OCc2ccccc2)ccc1O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.54
CA4 P22748 1/20 0.54
CA6 P23280 1/20 0.54
CA5A P35218 1/20 0.54
CA7 P43166 1/20 0.54
CA9 Q16790 1/20 0.54
CA14 Q9ULX7 1/20 0.54
CA5B Q9Y2D0 1/20 0.54
EGFR P00533 1/20 0.46
GAA P10253 3/20 0.45
TSHR P16473 2/20 0.45
BLM P54132 1/20 0.45
ALDH1A1 P00352 2/20 0.45
NFKB1 P19838 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CTSV O60911 1/20 0.45
CTSL P07711 1/20 0.45
TRPV1 Q8NER1 1/20 0.45
HSP90AA1 P07900 1/20 0.45
TTR P02766 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10832679 0.81 C5AR1 (0.51) GAAALDH1A1CTSVCTSLMEN1
SCHEMBL11453114 0.80 ALDH1A1 (0.56) GAAALDH1A1CTSLACHEKMT2A
SCHEMBL6412094 0.80 SMPD1 (0.54) ALDH1A1CTSVCTSLMEN1KMT2A
SCHEMBL3661649 0.80 TSHR (0.55) CA12CA4CA6CA5ACA7
SCHEMBL11454434 0.80 ALDH1A1 (0.54) CA12CA4CA6CA5ACA7
SCHEMBL6081043 0.79 ALDH1A1 (0.64) CA12CA4CA6CA5ACA7
SCHEMBL11471191 0.79 POLB (0.48) GAAALDH1A1TDP1MEN1KMT2A
SCHEMBL28532163 0.78 PTPN7 (0.58) EGFRGAABLMALDH1A1TRPV1
SCHEMBL62534 0.78 ALDH1A1 (0.59) ALDH1A1TDP1MEN1KMT2AMAPT
SCHEMBL11471660 0.77 ALDH1A1 (0.51) CA12CA9GAAALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957073-A2 MEDICINAL DRUG OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-08-20 EP disclosed
WO-2007066784-A2 DIARYLETHER DERIVATIVES AS ANTITUMOR AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-06-14 WO disclosed