SCHEMBL4716662

SCHEMBL4716662

CSC(=NC(=O)c1ccccc1)NCC(c1ccccc1)(c1ccc(F)cc1)c1cc(F)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DDR1 Q08345 4/20 0.40
P2RX1 P51575 1/20 0.39
CETP P11597 6/20 0.38
KCNH2 Q12809 3/20 0.38
SLC6A9 P48067 1/20 0.37
BCHE P06276 1/20 0.35
TACR1 P25103 1/20 0.35
TRPA1 O75762 2/20 0.35
CYP1A2 P05177 1/20 0.35
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL843676 0.80 CETP (0.57) CETPKCNH2
SCHEMBL843677 0.80 CETP (0.57) CETPKCNH2
SCHEMBL843674 0.80 CETP (0.57) CETPKCNH2
SCHEMBL843675 0.80 CETP (0.57) CETPKCNH2
SCHEMBL4969174 0.76 CETP (0.48) P2RX1CETPKCNH2SLC6A9TACR1
SCHEMBL4721472 0.74 CETP (0.41) P2RX1CETPKCNH2SLC6A9HTT
SCHEMBL4966775 0.73 CETP (0.43) P2RX1CETPKCNH2SLC6A9TACR1
SCHEMBL4967551 0.73 CETP (0.43) P2RX1CETPKCNH2SLC6A9TACR1
SCHEMBL4970220 0.73 CETP (0.43) P2RX1CETPKCNH2SLC6A9TACR1
SCHEMBL4971187 0.72 CETP (0.65) P2RX1CETPKCNH2SLC6A9TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951690-A1 HETEROCYCLIC CETP INHIBITORS Brystol-Myers Squibb Company (US) 2008-08-06 EP disclosed
WO-2007062342-A1 HETEROCYCLIC CETP INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-31 WO disclosed