SCHEMBL4717038

SCHEMBL4717038

O=C(O)CCc1c(F)ccc(F)c1F

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 6/20 0.49
FFAR4 Q5NUL3 4/20 0.49
KEAP1 Q14145 1/20 0.43
GPR17 Q13304 6/20 0.42
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29010008 0.88 FFAR4 (0.51) FFAR1FFAR4
SCHEMBL28805647 0.85 CES2 (0.40) FFAR1FFAR4GPR17CES2CES1
SCHEMBL19522398 0.85 GPR17 (0.55) FFAR1FFAR4KEAP1GPR17
SCHEMBL4718220 0.82 CES2 (0.38) FFAR1FFAR4GPR17CES2CES1
SCHEMBL27037031 0.81 FFAR1 (0.50) FFAR1FFAR4KEAP1GPR17CES2
SCHEMBL4714927 0.81 FFAR1 (0.59) FFAR1FFAR4KEAP1GPR17CES2
SCHEMBL29459948 0.78 AKR1B1 (0.43) FFAR4CES2CES1ALDH1A1
SCHEMBL909585 0.78 AKR1B1 (0.43) FFAR4CES2CES1ALDH1A1
SCHEMBL4717045 0.78 FFAR1 (0.49) FFAR1FFAR4KEAP1CES2CES1
SCHEMBL20889396 0.77 NPSR1 (0.44) FFAR1FFAR4KEAP1GPR17MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337517-B1 PYRIMIDINONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 2008-11-26 EP disclosed