SCHEMBL4717873

SCHEMBL4717873

NC1CC[C@H](S(=O)(=O)c2cc3c(cc2Cl)[nH]c(=O)c2[nH]ccc23)C1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.35
ROCK1 Q13464 2/20 0.34
AURKA O14965 1/20 0.30
TPX2 Q9ULW0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Butyric Acid SCHEMBL4161192 0.89 ROCK2 (0.33) ROCK2AURKATPX2
SCHEMBL4713961 0.83 PARG (0.38) ROCK2ROCK1
SCHEMBL3253927 0.79 CSNK2A2 (0.33)
SCHEMBL3253930 0.79 CSNK2A2 (0.33)
Hydrochloric Acid SCHEMBL3250727 0.79 CSNK2A2 (0.32)
Hydrochloric Acid SCHEMBL3250722 0.79 CSNK2A2 (0.32)
SCHEMBL4717883 0.76 GRIN2D (0.37)
Hydrochloric Acid SCHEMBL4161189 0.74 GPR17 (0.32)
Butyric Acid SCHEMBL4167771 0.73 BRAF (0.33) ROCK2
Butyric Acid SCHEMBL4166107 0.73 BRAF (0.33) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-A1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PIERRE FABRE MEDICAMENT (FR) 2008-03-19 EP claimed
WO-2007003611-A1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PIERRE FABRE MEDICAMENT (FR) 2007-01-11 WO claimed