SCHEMBL47183

SCHEMBL47183

C/C=C(/NC(CO)CO)c1ccc2c(c1)C(C)(C)CC(c1cccc(N3CCOCC3)c1)N2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.34
CYP3A4 P08684 3/20 0.34
PLOD2 O00469 2/20 0.33
PLOD3 O60568 2/20 0.33
PLOD1 Q02809 2/20 0.33
KIF11 P52732 3/20 0.32
KMO O15229 1/20 0.31
CYP2C9 P11712 2/20 0.31
F10 P00742 2/20 0.31
F11 P03951 2/20 0.31
F7 P08709 2/20 0.31
KCNQ3 O43525 1/20 0.31
KCNQ2 O43526 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP19A1 P11511 1/20 0.31
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
MEN1 O00255 1/20 0.30
PSMD14 O00487 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15760093 0.89 CYP2C19 (0.35) CYP2C19CYP3A4PLOD2PLOD3PLOD1
SCHEMBL45003 0.89 F10 (0.39) CYP2C19CYP3A4PLOD2PLOD3PLOD1
SCHEMBL15751977 0.83 KDM4E (0.38) CYP2C19CYP3A4MEN1ALDH1A1MAPT
SCHEMBL45312 0.82 F10 (0.47) CYP2C19CYP3A4PLOD2PLOD3PLOD1
SCHEMBL41549 0.81 KMO (0.52) CYP2C19CYP3A4PLOD2PLOD3PLOD1
SCHEMBL45257 0.81 PRMT5 (0.44) CYP2C19PLOD2PLOD3PLOD1MEN1
SCHEMBL45781 0.81 F10 (0.45) CYP2C19CYP3A4PLOD2PLOD3PLOD1
SCHEMBL11026483 0.81 F10 (0.45) CYP2C19CYP3A4PLOD2PLOD3PLOD1
SCHEMBL45394 0.80 PRKD1 (0.40) CYP2C19CYP3A4PLOD2PLOD3PLOD1
SCHEMBL11025709 0.80 F7 (0.44) CYP2C19CYP3A4PLOD2PLOD3PLOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001020-A1 NOVEL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-05 WO disclosed