SCHEMBL4718800

SCHEMBL4718800

NC(=O)c1ccc2nc3[nH]cccc-3c2c1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 17/20 0.50
PKN1 Q16512 1/20 0.43
PKN2 Q16513 1/20 0.43
IP6K1 Q92551 1/20 0.42
CHEK1 O14757 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4088326 0.89 CHEK2 (0.44) CHEK2PKN1PKN2CHEK1
SCHEMBL15534807 0.79 CHEK2 (0.46) CHEK2PKN1PKN2
SCHEMBL1180188 0.71 NPC1 (0.47)
Hydrochloric Acid SCHEMBL4972256 0.69 GRM2 (0.44) CHEK2PKN2CHEK1
SCHEMBL24976057 0.69 IP6K1 (0.48) CHEK2IP6K1
SCHEMBL31428714 0.69 IP6K1 (0.48) CHEK2IP6K1
SCHEMBL1181806 0.68 ACHE (0.41)
SCHEMBL4507302 0.68 CHEK2 (0.59) CHEK2PKN1PKN2CHEK1
SCHEMBL31428846 0.67 IP6K1 (0.46) CHEK2PKN2IP6K1CHEK1
SCHEMBL24976114 0.67 IP6K1 (0.46) CHEK2PKN2IP6K1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940840-A1 6-HETEROARYLPYRIDOINDOLONE DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC USE THEREOF Sanofi-Aventis (FR) 2008-07-09 EP disclosed
WO-2007045758-A1 6-HETEROARYLPYRIDOINDOLONE DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC USE THEREOF SANOFI AVENTIS (FR) 2007-04-26 WO disclosed