SCHEMBL4720180

SCHEMBL4720180

O=S(=O)(CCCC(O)c1ncccn1)N1CCN(c2ccc(OCC(F)(F)F)cn2)CC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 16/20 0.46
CYP3A4 P08684 1/20 0.44
MMP13 P45452 1/20 0.44
KDM4E B2RXH2 2/20 0.41
HSD17B10 Q99714 1/20 0.41
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
MMP7 P09237 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3939247 0.81 CYP3A4 (0.53) GPR119CYP3A4MMP13KDM4EALDH1A1
SCHEMBL13941032 0.79 CYP3A4 (0.56) GPR119CYP3A4MMP13KDM4EALDH1A1
SCHEMBL5765295 0.79 GPR119 (0.44) GPR119KDM4E
SCHEMBL3936734 0.79 CYP3A4 (0.51) GPR119CYP3A4MMP13KDM4EALDH1A1
SCHEMBL5763519 0.77 GPR119 (0.44) GPR119KDM4E
SCHEMBL3942539 0.76 CYP3A4 (0.46) GPR119CYP3A4MMP13KDM4EALDH1A1
SCHEMBL3940021 0.76 CYP3A4 (0.52) GPR119CYP3A4MMP13MMP7
SCHEMBL3943472 0.75 GAA (0.46) GPR119KDM4E
SCHEMBL13923649 0.75 CYP3A4 (0.80) GPR119CYP3A4MMP13MMP7
SCHEMBL3940017 0.74 CYP3A4 (0.72) GPR119CYP3A4MMP13MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644340-B1 N-[({'4-SUBSTITUTED PIPERAZINE-1-YL}SULFONYLMETHYL)ALKYL]-N-HYDROXYFORMAMIDE COMPOUNDS AS METALLOPROTEINASE INHIBITORS ASTRAZENECA AB (SE) 2008-11-12 EP disclosed