SCHEMBL4720518

SCHEMBL4720518

COc1cc(OC)cc(-c2cc(-c3cc(N4CCC(O)C4)ccc3C(F)(F)F)c(OC)c3c2CCC3)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 0.35
ICAM1 P05362 1/20 0.35
ITGAL P20701 1/20 0.35
SOS1 Q07889 2/20 0.34
P2RX7 Q99572 1/20 0.34
ABL1 P00519 1/20 0.34
NOTUM Q6P988 1/20 0.33
LRRK2 Q5S007 1/20 0.33
AR P10275 1/20 0.33
CDK1 P06493 1/20 0.33
CDK2 P24941 1/20 0.33
F10 P00742 2/20 0.33
HSD11B1 P28845 2/20 0.33
F2 P00734 1/20 0.33
S1PR1 P21453 1/20 0.33
ACACB O00763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720516 1.00 ITGB2 (0.35) ITGB2ICAM1ITGALSOS1P2RX7
SCHEMBL4720760 0.91 CDK1 (0.35) ITGB2ICAM1ITGALSOS1P2RX7
SCHEMBL4720758 0.91 CDK1 (0.35) ITGB2ICAM1ITGALSOS1P2RX7
SCHEMBL4720319 0.89 ITGB2 (0.36) ITGB2ICAM1ITGALABL1LRRK2
SCHEMBL4720326 0.89 ITGB2 (0.36) ITGB2ICAM1ITGALABL1LRRK2
SCHEMBL4719067 0.87 ITGB2 (0.35) ITGB2ICAM1ITGALSOS1P2RX7
SCHEMBL4719061 0.87 ITGB2 (0.35) ITGB2ICAM1ITGALSOS1P2RX7
SCHEMBL4721675 0.84 CDK1 (0.38) ITGB2ICAM1ITGALSOS1ABL1
SCHEMBL4721666 0.84 CDK1 (0.38) ITGB2ICAM1ITGALSOS1ABL1
SCHEMBL4721351 0.80 P2RX7 (0.34) ITGB2ICAM1ITGALSOS1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed