SCHEMBL4720527

SCHEMBL4720527

CNC(=O)CCCNc1ccc(C(F)(F)F)c(-n2nc(-c3cc(OC)cc(OC)c3)c3cc(C)[nH]c3c2=O)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD O00767 4/20 0.34
FPR1 P21462 2/20 0.33
FPR2 P25090 2/20 0.33
ALDH1A1 P00352 2/20 0.32
CARM1 Q86X55 1/20 0.31
MAPT P10636 1/20 0.31
ALPG P10696 1/20 0.31
HPGD P15428 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
MAPK10 P53779 1/20 0.31
HSD17B10 Q99714 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
KDM4E B2RXH2 1/20 0.30
HSD17B1 P14061 1/20 0.30
HSD17B2 P37059 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719300 0.89 BRD4 (0.35) SCDFPR1FPR2ALDH1A1TSHR
SCHEMBL4724683 0.85 SCD (0.33) SCDFPR1FPR2ALDH1A1MAPT
SCHEMBL4720549 0.84 SCD (0.33) SCDFPR1FPR2MAPTTP53
SCHEMBL4723187 0.83 MAPT (0.34) SCDFPR1FPR2MAPTTP53
SCHEMBL4724929 0.82 SCD (0.32) SCDFPR1FPR2KDM4EHSD17B1
SCHEMBL4719384 0.81 MAPT (0.34) SCDFPR1FPR2MAPTTP53
SCHEMBL4722630 0.79 F10 (0.31) SCDFPR1FPR2KDM4ERXFP1
SCHEMBL4719755 0.78 MAPT (0.35) SCDFPR1FPR2MAPTTP53
SCHEMBL14101715 0.76 AR (0.38) ALDH1A1MAPTHPGDNPSR1TDP1
SCHEMBL4765721 0.75 PDE4A (0.36) SCDMAPTTP53TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed